Compound 5h , in particular , displayed the most potent inhibitory activity , with a K i value of 0.006 mM.
This potency was 65-fold higher than the potency of the lead compound 4 ( K i ¼ 0.39 mM ) .
Compound 5h , in particular , displayed the most potent inhibitory activity , with a K i value of 0.006 mM.
This potency was 65-fold higher than the potency of the lead compound 4 ( K i ¼ 0.39 mM ) .